Synthesis of the Benzo-fused Indolizidine Alkaloid Mimics
نویسندگان
چکیده
منابع مشابه
Synthesis of the Benzo-fused Indolizidine Alkaloid Mimics
A general synthesis of various benzo-fused indolizidine alkaloid mimics has been developed. The indolizidine derivatives 8 were prepared via heteroaryl Grignard addition to N-acylpyridinium salts followed by an intramolecular Heck cyclization. Further substitution reactions were developed to demonstrate that heterocycles 8 are good scaffolds for chemical library preparation.
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ژورنال
عنوان ژورنال: Beilstein Journal of Organic Chemistry
سال: 2007
ISSN: 1860-5397
DOI: 10.1186/1860-5397-3-42